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Accueil > Productions scientifiques

2014

publié le , mis à jour le

1. Revues à comité de lecture

Asgatay S., Champion C., Marloie G., Drujon T., Senamaud-Beaufort C., Ceccaldi A., Erdmann A., Rajavelu A., Schambel P., Jeltsch A., Lequin O., Karoyan P., Arimondo PB., Guianvarc’h D., Synthesis and Evaluation of Analogues of N-Phthaloyl-l-tryptophan (RG108) as Inhibitors of DNA Methyltransferase 1.,J Med Chem, 2014, 57(2):421-34

D’Ambrosio K., Lopez M., A Dathan N., Ouahrani-Bettache S.,Köhler S., Ascione G., Maria Monti S., Winum JY. and De Simone G., Structural basis for the rational design of new anti-Brucella agents : the crystal structure of the C366S mutant of HDH from Brucella suis, Biochimie, 2014, 97, 114-120

Erdmann A., Halby L., Cantagrel F., Sautel F., Massiot G., Arimondo PB., Alternative synthetic route to annulated diaminopyrimidines,Tet. Lett., 2014, 55 (29), 3901-3904

Guianvarc’h D., Arimondo PB., Challenges in developing novel DNA methyltransferases inhibitors for cancer therapy, Future Medicinal Chemistry, 2014, 6(11) 1237-40

Jiang Y., Zeng KW., David B., Massiot G., Constituents of Vigna angularis and their in vitro anti-inflammatory activity, Phytochemistry, 2014, 107, 111-118

Khouni L., Long C., Haba H., Molinier N. and Benkhaled M., Anthranilic Acid Derivatives and Other Components from Ononis pusilla, Nat. Prod. Comm., 2014, 9(8), 1159-1162

Lopez M., Laurent F., Bornaghi LF. and Poulsen SA., Synthesis of sulfomanide-conjugated glycosyl-amino acid building blocks, Carbohydrate Res., 2014, 386, 78-85

Moison C., Assemat F., Daunay A., Tost J., Guiyesse-Peugeot AL., ArimondoPB., Synergistic chromatin repression of the tumor suppressor gene RARB in human prostate cancers,Epigenetics,2014 9(4), 477-482

Pouny I., Batut M., Vendier L.,David B., Yi S., Sautel F., Arimondo PB., Massiot G., Cytisine-like alkaloids from Ormosia hosiei Hemsley & E. H. Wilson, Phytochemistry, 2014, Volume 107, Pages 97-101

Rilova E., Erdmann A., Gros C., Masson V., Aussagues Y., Poughon-Cassabois V., Rajavelu A., Jeltsch A., Menon Y., Novosad N., Gregoire JM.,Vispé S., Schambel P., Ausseil A., Sautel F., Arimondo PB. andCantagrel F., Design, synthesis and biological evaluation of 4-amino-N-(4-aminophenyl)-benzamides analogues of quinoline-based SGI-1027 as inhibitors of DNA methylation, ChemMedChem, 2014, 9(3), 590-601

Rotili D., Tarantino D., Marrocco B., Gros C., Masson V., Poughon V., Ausseil F., Chang Y., Labella D., Cosconati S., Di Maro S., Novellino E., Schnekenburger M., Grandjenette C., Bouvy C., Diederich M., Cheng X., Arimondo PB.,Mai A., Properly Substituted Analogues of BIX-01294 Lose Inhibition of G9a Histone Methyltransferase and Gain Selective Anti-DNA Methyltransferase 3A Activity., PLoS One.,2014, 29(5):e96941

Turtaut F., Lopez M., Ouahrani-Bettache S., Köhler S., Winum JY., Oxo- and thiooxo-imidazo[1,5-c]pyrimidine molecule library : beyond their interest in inhibition of Brucella suis histidinol dehydrogenase, a powerful protection tool in the synthesis of histidine analogues, Bioorg. Med. Chem. Lett., in press

Valente S., Yiwei L., Schnekenburger M., Zwergel C., Cosconati S., Gros C., Tardugno M., Labella D., Florean C., Minden S., Hashimoto H., Chang Y., Zhang X., Kirsch G., Novellino E., Arimondo PB., Miele E., Ferretti E., Gulino A., Diederich M., Cheng X., Mai A., Selective Non-Nucleoside Inhibitors of Human DNA Methyltransferases Active in Cancer Including Cancer Stem Cells.,J. Med. Chem.,2014, 57, 701−713

2. Ouvrages, chapitres d’ouvrages

Arimondo PB., Guilbaud N., Bailly C., A new generation of cell-targeted drugs for cancer treatment.Chapter Book in Cancer Drug Design and Discovery, 2014, pp 177-191. Editor Stephen Neidle, Elsevier

David B., Ausseil F., High Throughput Screening of Vegetal Natural Substances, Handbook of Chemical and Biological Plant Analytical Methods, edited by Kurt Hostettmann, Shilin Chen, Andrew Marston and Hermann Stuppner, Chichester, UK, John Wiley & Sons, Ltd, pp 987-1010.

Moison C., Assemat F., Daunay A., Arimondo PB., and Tost J., Single nucleotide resolution methylation analysis of ChIP products,Methods in Molecular Biology, Pyrosequencing, Springer, in press